ROS1 — Targeted Therapies, Trials & Pipeline
ROS1 rearrangements are a rare but highly targetable oncogenic driver in NSCLC.
Approved drugs targeting ROS1
brigatinib
·
ceritinib
·
crizotinib
·
Entrectinib
·
Repotrectinib
·
Taletrectinib
·
Zidesamtinib
Investigational pipeline agents
APG-2449