FLT3 — Targeted Therapies, Trials & Pipeline
FLT3-ITD and TKD mutations are adverse-risk drivers in AML, now targeted by FLT3 inhibitors.
Approved drugs targeting FLT3
gilteritinib
·
midostaurin
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ponatinib
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quizartinib
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Sorafenib
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Sunitinib
Investigational pipeline agents
BMF-500
·
Emavusertib
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Tuspetinib
·
Zotiraciclib
Landmark trials
RATIFY